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Скачать или смотреть Antidiabetic drugs pharmacology, DDP 4 inhibitors pharmacology, clinical pharmacology diabetes

  • pharmacy by asim
  • 2025-03-22
  • 232
Antidiabetic drugs pharmacology, DDP 4 inhibitors pharmacology, clinical pharmacology diabetes
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Описание к видео Antidiabetic drugs pharmacology, DDP 4 inhibitors pharmacology, clinical pharmacology diabetes

💊 Dipeptidyl Peptidase-4 (DPP-4) inhibitors are a class of oral anti-diabetic drugs that work by enhancing the body’s natural incretin hormones, which are involved in glucose homeostasis. DPP-4 inhibitors enhance postprandial insulin release and decrease glucagon levels, leading to better glycemic control. They are primarily used in the treatment of Type 2 diabetes mellitus (T2DM).

✅ Mechanism: Inhibit DPP-4 enzyme → Increase GLP-1 & GIP → Enhance insulin secretion & suppress glucagon.
✅ Indications: Type 2 Diabetes Mellitus (Not used in Type 1 DM).
✅ Drugs in Class: Sitagliptin, Linagliptin, Saxagliptin, Alogliptin, Vildagliptin.
✅ Dosing: Usually once daily; renal adjustment needed except for linagliptin.
✅ Weight Effects: Weight-neutral (unlike GLP-1 RAs, which cause weight loss).
✅ Side Effects: Nasopharyngitis, headache, joint pain, pancreatitis (rare).
✅ Drug Interactions: Saxagliptin → Metabolized by CYP3A4 → Risk of interactions.
✅ Heart Failure: Saxagliptin may increase heart failure risk (caution in CHF patients).
#diabetes #DDP4inhibitors #pharmcologylectures #clinicalpharmacology

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Chapters:
0:00 - DPP-4 inhibitors pharmacology
0:31 - DPP-4 inhibitors clinical pharmacology
0:39 - DPP-4 inhibitors renal dose adjustments
1:15 - DPP-4 inhibitors and hypoglycemia risk
1:41 - DPP-4 inhibitors and heart failure
2:08 - DPP-4 inhibitors and pancreatitis risk
2:29 - DPP-4 inhibitors combination therapy
2:59 - DPP-4 inhibitors and weight loss
3:33 - DPP-4 inhibitors clinical pharmacology summary

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