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Скачать или смотреть Antidiabetic drugs pharmacology, SGLT 2 inhibitors pharmacology, clinical pharmacology diabetes

  • pharmacy by asim
  • 2025-03-19
  • 303
Antidiabetic drugs pharmacology, SGLT 2 inhibitors pharmacology, clinical pharmacology diabetes
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💊 Sodium-glucose co-transporter 2 inhibitors also known as SGLT-2 inhibitors are a class of oral antidiabetic agents that reduce blood glucose levels by promoting the excretion of glucose in the urine. They primarily act in the proximal renal tubules to block glucose reabsorption, leading to glucosuria.

✅ SGLT-2 inhibitors (e.g., empagliflozin, dapagliflozin, canagliflozin) lower blood glucose by increasing glucose excretion in the urine.
✅ Provide cardiovascular and renal protection beyond glucose control.
✅ Reduce weight and blood pressure via osmotic diuresis.
✅ Common side effects: Genital and urinary tract infections, dehydration, hypotension.
✅ Rare but serious risks: Euglycemic diabetic ketoacidosis (DKA), lower limb amputations (with canagliflozin).
✅ Should not be used in eGFR less than 30 mL/min (except dapagliflozin for CKD less than 25 mL/min).
✅ Should be stopped before surgery to reduce DKA risk.
#sglt2 #diabetes #antidiabetic #pharamacologylectures #clinicalpharmacology

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Chapters:
0:00 - SGLT-2 inhibitors pharmacology
0:23 - SGLT-2 inhibitors clinical pharmacology
0:31 - SGLT-2 inhibitors and DKA risk
1:01 - SGLT-2 inhibitors and cardiovascular benefits
1:29 - SGLT-2 inhibitors and genital infections
1:49 - SGLT-2 inhibitors and weight loss
2:06 - SGLT-2 inhibitors and renal impairment
2:27 - SGLT-2 inhibitors summary

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